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Small molecule ERK5 kinase inhibitors paradoxically activate ERK5 signalling: be careful what you wish for…

ERK5 is a protein kinase that also contains a nuclear localisation signal and a transcriptional transactivation domain. Inhibition of ERK5 has therapeutic potential in cancer and inflammation and this has prompted the development of ERK5 kinase inhibitors (ERK5i). However, few ERK5i programmes have...

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Kaydedildi:
Detaylı Bibliyografya
Yayımlandı:Biochem Soc Trans
Asıl Yazarlar: Cook, Simon J., Tucker, Julie A., Lochhead, Pamela A.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Portland Press Ltd. 2020
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC7609025/
https://ncbi.nlm.nih.gov/pubmed/32915196
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BST20190338
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