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The Development and Validation of a Novel “Dual Cocktail” Probe for Cytochrome P450s and Transporter Functions to Evaluate Pharmacokinetic Drug-Drug and Herb-Drug Interactions

This study was designed to develop and validate a 10 probe drug cocktail named “Dual Cocktail”, composed of caffeine (Cyp1a2 in rat and CYP1A2 in human, 1 mg/kg), diclofenac (Cyp2c11 in rat and CYP2C9 in human, 2 mg/kg), omeprazole (Cyp2c11 in rat and CYP2C19 in human, 2 mg/kg), dextromethorphan (Cy...

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Bibliografski detalji
Izdano u:Pharmaceutics
Glavni autori: Kwon, Mihwa, Jeon, Ji-Hyeon, Choi, Min-Koo, Song, Im-Sook
Format: Artigo
Jezik:Inglês
Izdano: MDPI 2020
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7600799/
https://ncbi.nlm.nih.gov/pubmed/33007943
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics12100938
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