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The dual HDAC-PI3K inhibitor CUDC-907 displays single-agent activity and synergizes with PARP inhibitor olaparib in small cell lung cancer

BACKGROUND: Small cell lung cancer (SCLC) is a deadly neuroendocrine tumor with limited therapeutic options. Recent data suggest that histone deacetylases (HDACs) and the phosphatidylinositol 3-kinase (PI3K) pathway play essential roles in SCLC cell proliferation and survival. METHODS: The inhibitio...

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Detalhes bibliográficos
Publicado no:J Exp Clin Cancer Res
Main Authors: Ma, Liying, Bian, Xing, Lin, Wenchu
Formato: Artigo
Idioma:Inglês
Publicado em: BioMed Central 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7568419/
https://ncbi.nlm.nih.gov/pubmed/33069237
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/s13046-020-01728-2
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