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Ponatinib and other CML Tyrosine Kinase Inhibitors in Thrombosis

Abl1 kinase has important biological roles. The Bcr-Abl1 fusion protein creates undesired kinase activity and is pathogenic in 95% of chronic myeloid leukemia (CML) and 30% of acute lymphoblastic leukemia (ALL) patients. Targeted therapies to these diseases are tyrosine kinase inhibitors. The extent...

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Dades bibliogràfiques
Publicat a:Int J Mol Sci
Autors principals: Zeng, Peng, Schmaier, Alvin
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7555546/
https://ncbi.nlm.nih.gov/pubmed/32911643
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms21186556
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