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CYP1A1 and Cnr nitroreductase bioactivated niclosamide in vitro

Niclosamide produces genotoxic effects, such as point mutations in Salmonella sp., sperm-head abnormalities in mice and clastogenic effects in human lymphocytes in vitro and in vivo. As cytochrome P450 could be involved in the bioactivation of niclosamide, we investigated which subfamily was involve...

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Bibliografiske detaljer
Udgivet i:Mutagenesis
Main Authors: Beristain-Castillo, Evelyn, Martínez-Vázquez, Mariano, Camacho-Carranza, Rafael, Espinosa-Aguirre, Javier J.
Format: Artigo
Sprog:Inglês
Udgivet: Oxford University Press 2013
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7539354/
https://ncbi.nlm.nih.gov/pubmed/23956140
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/mutage/get043
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