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Discovery of gramicidin A analogues with altered activities by multidimensional screening of a one-bead-one-compound library

Gramicidin A (1) is a peptide antibiotic that disrupts the transmembrane ion concentration gradient by forming an ion channel in a lipid bilayer. Although long used clinically, it is limited to topical application because of its strong hemolytic activity and mammalian cytotoxicity, likely arising fr...

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Bibliografiska uppgifter
I publikationen:Nat Commun
Huvudupphovsmän: Takada, Yuri, Itoh, Hiroaki, Paudel, Atmika, Panthee, Suresh, Hamamoto, Hiroshi, Sekimizu, Kazuhisa, Inoue, Masayuki
Materialtyp: Artigo
Språk:Inglês
Publicerad: Nature Publishing Group UK 2020
Ämnen:
Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC7531004/
https://ncbi.nlm.nih.gov/pubmed/33004797
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41467-020-18711-2
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