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Metabolism of a Bioorthogonal PET Tracer Candidate [(19)F/(18)F]SiFA-Tetrazine in Mouse Liver Microsomes: Biotransformation Pathways and Defluorination Investigated by UHPLC-HRMS
[Image: see text] Organofluorosilicon based (18)F-radiolabeling is an efficient method for incorporating fluorine-18 into (18)F-radiopharmaceuticals for positron emission tomography (PET) by (19)F/(18)F isotopic exchange (IE). The first PET radiopharmaceutical, (18)F-SiFAlin-TATE, radiolabeled with...
Salvato in:
| Pubblicato in: | Mol Pharm |
|---|---|
| Autori principali: | , , , |
| Natura: | Artigo |
| Lingua: | Inglês |
| Pubblicazione: |
American Chemical
Society
2020
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| Accesso online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7497667/ https://ncbi.nlm.nih.gov/pubmed/32539414 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.molpharmaceut.0c00523 |
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