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Characterization of platinum(II) complexes exhibiting inhibitory activity against the 20S proteasome

Proteasome inhibitors are useful for biochemical research and clinical treatment. In our previous study, we reported that the 4N-coordinated platinum complexes with anthracenyl ring and heterocycle exhibited proteasome-inhibitory activity. In the present study, the structure–activity relationships a...

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Pubblicato in:R Soc Open Sci
Autori principali: Kiwada, Tatsuto, Katakasu, Hiromu, Okumura, Serina, Odani, Akira
Natura: Artigo
Lingua:Inglês
Pubblicazione: The Royal Society 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7481701/
https://ncbi.nlm.nih.gov/pubmed/32968518
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1098/rsos.200545
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