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Development of Alkyne-Containing Pyrazolopyrimidines To Overcome Drug Resistance of Bcr-Abl Kinase

Despite the success of imatinib at inhibiting Bcr-Abl and treating chronic myelogenous leukemia (CML), resistance to the therapy occurs over time in patients. In particular, the resistance to imatinib caused by the gatekeeper mutation T315I in Bcr-Abl remains a challenge in the clinic. Inspired by t...

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Bibliografische gegevens
Gepubliceerd in:J Med Chem
Hoofdauteurs: Liu, Xu, Kung, Alvin, Malinoski, Brock, Prakash, G. K. Surya, Zhang, Chao
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: 2015
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Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7475166/
https://ncbi.nlm.nih.gov/pubmed/26562217
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b01125
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