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Design of drug-like hepsin inhibitors against prostate cancer and kidney stones

Hepsin, a transmembrane serine protease abundant in renal endothelial cells, is a promising therapeutic target against several cancers, particularly prostate cancer. It is involved in the release and polymerization of uromodulin in the urine, which plays a role in kidney stone formation. In this wor...

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Publicat a:Acta Pharm Sin B
Autors principals: Blay, Vincent, Li, Mu-Chun, Ho, Sunita P., Stoller, Mashall L., Hsieh, Hsing-Pang, Houston, Douglas R.
Format: Artigo
Idioma:Inglês
Publicat: Elsevier 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7452031/
https://ncbi.nlm.nih.gov/pubmed/32874830
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.apsb.2019.09.008
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