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Rigid Scaffolds: Synthesis of 2,6‐Bridged Piperazines with Functional Groups in all three Bridges

The activity of pharmacologically active compounds can be increased by presenting a drug in a defined conformation, which fits exactly into the binding pocket of its target. Herein, the piperazine scaffold was conformationally restricted by substituted C(2)‐ or C(3)‐bridges across the 2‐ and 6‐posit...

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Bibliografische gegevens
Gepubliceerd in:ChemistryOpen
Hoofdauteurs: Gao, Donglin, Penno, Christian, Wünsch, Bernhard
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: John Wiley and Sons Inc. 2020
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Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7450790/
https://ncbi.nlm.nih.gov/pubmed/32884883
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/open.202000188
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