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A Macromolecular Janus Kinase (JAK) Inhibitor Prodrug Effectively Ameliorates Dextran Sulfate Sodium-induced Ulcerative Colitis in Mice

BACKGROUND: Tofacitinib (Tofa) has been approved for moderately to severely active ulcerative colitis (UC). To improve its therapeutic efficacy and limit dose-dependent toxicity, we developed a macromolecular prodrug of Tofa (P-Tofa). If the prodrug design improves the potency and duration of Tofa t...

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Détails bibliographiques
Publié dans:Pharm Res
Auteurs principaux: Zhao, Gang, Wei, Xin, Wu, Jianbo, Eichele, Derrick D, Lele, Subodh M., Yang, Libin, Zhang, Fan, Wang, Dong
Format: Artigo
Langue:Inglês
Publié: 2019
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7433013/
https://ncbi.nlm.nih.gov/pubmed/30859327
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11095-019-2587-6
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