Caricamento...

In vitro and in vivo evaluation of the antimalarial MMV665831 and structural analogs

Antimalarial candidates possessing novel mechanisms of action are needed to control drug resistant Plasmodium falciparum. We were drawn to Malaria Box compound 1 (MMV665831) by virtue of its excellent in vitro potency, and twelve analogs were prepared to probe its structure-activity relationship. Mo...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Pubblicato in:Bioorg Med Chem Lett
Autori principali: Ding, Sha, Fike, Katherine R., Klemba, Michael, Carlier, Paul R.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2020
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7422479/
https://ncbi.nlm.nih.gov/pubmed/32738996
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2020.127348
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !