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Synthesis, docking study and biological evaluation of ᴅ-fructofuranosyl and ᴅ-tagatofuranosyl sulfones as potential inhibitors of the mycobacterial galactan synthesis targeting the galactofuranosyltransferase GlfT2

A series of ten novel ᴅ-fructofuranosyl and ᴅ-tagatofuranosyl sulfones bearing a 1-O-phosphono moiety and three different substituents at C-2 has been prepared. Due to the structural similarities of these scaffolds to the native substrate of mycobacterial galactofuranosyltransferase GlfT2 in the tra...

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Библиографические подробности
Опубликовано в: :Beilstein J Org Chem
Главные авторы: Baráth, Marek, Jakubčinová, Jana, Konyariková, Zuzana, Kozmon, Stanislav, Mikušová, Katarína, Bella, Maroš
Формат: Artigo
Язык:Inglês
Опубликовано: Beilstein-Institut 2020
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC7404141/
https://ncbi.nlm.nih.gov/pubmed/32802202
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.16.152
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