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Macrocycle Cell Permeability Measured by Solvation Free Energies in Polar and Apolar Environments

[Image: see text] The relation of surface polarity and conformational preferences is decisive for cell permeability and thus bioavailability of macrocyclic drugs. Here, we employ grid inhomogeneous solvation theory (GIST) to calculate solvation free energies for a series of six macrocycles in water...

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Detalhes bibliográficos
Publicado no:J Chem Inf Model
Main Authors: Kamenik, Anna S., Kraml, Johannes, Hofer, Florian, Waibl, Franz, Quoika, Patrick K., Kahler, Ursula, Schauperl, Michael, Liedl, Klaus R.
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2020
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7388155/
https://ncbi.nlm.nih.gov/pubmed/32551643
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jcim.0c00280
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