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Activity of Epigenetic Inhibitors against Plasmodium falciparum Asexual and Sexual Blood Stages

Earlier genetic and inhibitor studies showed that epigenetic regulation of gene expression is critical for malaria parasite survival in multiple life stages and a promising target for new antimalarials. We therefore evaluated the activity of 350 diverse epigenetic inhibitors against multiple stages...

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Publicado en:Antimicrob Agents Chemother
Autores principales: Vanheer, Leen N., Zhang, Hao, Lin, Gang, Kafsack, Björn F. C.
Formato: Artigo
Lenguaje:Inglês
Publicado: American Society for Microbiology 2020
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7318029/
https://ncbi.nlm.nih.gov/pubmed/32366713
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.02523-19
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