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Protein Binding Pocket Optimization for Virtual High-Throughput Screening (vHTS) Drug Discovery

[Image: see text] The virtual high-throughput screening (vHTS) approach has been widely used for large database screening to identify potential lead compounds for drug discovery. Due to its high computational demands, docking that allows receptor flexibility has been a challenging problem for virtua...

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Detalhes bibliográficos
Publicado no:ACS Omega
Main Authors: Gazgalis, Dimitris, Zaka, Mehreen, Abbasi, Bilal Haider, Logothetis, Diomedes E., Mezei, Mihaly, Cui, Meng
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2020
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7315428/
https://ncbi.nlm.nih.gov/pubmed/32596567
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsomega.0c00522
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