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Effect of P-glycoprotein (P-gp) Inducers on Exposure of P-gp Substrates: Review of Clinical Drug–Drug Interaction Studies

Understanding transporter-mediated drug–drug interactions (DDIs) for investigational agents is important during drug development to assess DDI liability, its clinical relevance, and to determine appropriate DDI management strategies. P-glycoprotein (P-gp) is an efflux transporter that influences the...

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Bibliografiske detaljer
Udgivet i:Clin Pharmacokinet
Main Authors: Elmeliegy, Mohamed, Vourvahis, Manoli, Guo, Cen, Wang, Diane D.
Format: Artigo
Sprog:Inglês
Udgivet: Springer International Publishing 2020
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7292822/
https://ncbi.nlm.nih.gov/pubmed/32052379
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s40262-020-00867-1
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