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Computational Simulations to Guide Enzyme-Mediated Prodrug Activation
Prodrugs are designed to improve pharmaceutical/biopharmaceutical characteristics, pharmacokinetic/pharmacodynamic properties, site-specificity, and more. A crucial step in successful prodrug is its activation, which releases the active parent drug, exerting a therapeutic effect. Prodrug activation...
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| Publicado no: | Int J Mol Sci |
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| Main Authors: | , , |
| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado em: |
MDPI
2020
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| Assuntos: | |
| Acesso em linha: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7279318/ https://ncbi.nlm.nih.gov/pubmed/32443905 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms21103621 |
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