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Characterisation of mexiletine’s translational therapeutic index for suppression of ischaemia-induced ventricular fibrillation in the rat isolated heart

The ‘translational therapeutic index’ (TTI) is a drug’s ratio of nonclinical threshold dose (or concentration) for significant benefit versus threshold for adversity. In early nonclinical research, discovery and safety studies are normally undertaken separately. Our aim was to evaluate a novel integ...

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Détails bibliographiques
Publié dans:Sci Rep
Auteurs principaux: Hesketh, Louise M., Wilder, Catherine D. E., Ranadive, Niraja N., Lytra, Georgia, Qazimi, Patrisia, Munro, Jade S., Ahdi, Nakita, Curtis, Michael J.
Format: Artigo
Langue:Inglês
Publié: Nature Publishing Group UK 2020
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7242333/
https://ncbi.nlm.nih.gov/pubmed/32439959
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-020-65190-y
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