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Total Synthesis of (+)-Granatumine A and Related Bislactone Limonoid Alkaloids via a Pyran to Pyridine Interconversion

We report the first total synthesis of (+)-granatumine A, a limonoid alkaloid with PTP1B inhibitory activity, in ten steps. Over the course of this study, two key methodological advances were made: a cost-effective procedure for ketone α,β-dehydrogenation using allyl-Pd catalysis, and a Pd-catalyzed...

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Pubblicato in:J Am Chem Soc
Autori principali: Schuppe, Alexander W., Zhao, Yizhou, Liu, Yannan, Newhouse, Timothy R.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7192014/
https://ncbi.nlm.nih.gov/pubmed/31117671
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.9b04508
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