Cargando...

Fedratinib in myelofibrosis

Following the discovery of the JAK2V617F mutation in myeloproliferative neoplasms in 2005, fedratinib was developed as a small molecular inhibitor of JAK2. It was optimized to yield low-nanomolar activity against JAK2 (50% inhibitory concentration = 3 nM) and was identified to be selective for JAK2...

Descripción completa

Guardado en:
Detalles Bibliográficos
Publicado en:Blood Adv
Autores principales: Mullally, Ann, Hood, John, Harrison, Claire, Mesa, Ruben
Formato: Artigo
Lenguaje:Inglês
Publicado: American Society of Hematology 2020
Materias:
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7189288/
https://ncbi.nlm.nih.gov/pubmed/32343799
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/bloodadvances.2019000954
Etiquetas: Agregar Etiqueta
Sin Etiquetas, Sea el primero en etiquetar este registro!