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Nickel-Catalyzed Conversion of Amides to Carboxylic Acids

We report the conversion of amides to carboxylic acids using nonprecious metal catalysis. The methodology strategically employs a nickel-catalyzed esterification using 2-(trimethylsilyl)-ethanol, followed by a fluoride-mediated deprotection in a single-pot operation. This approach circumvents cataly...

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Publicat a:Org Lett
Autors principals: Knapp, Rachel R., Bulger, Ana S., Garg, Neil K.
Format: Artigo
Idioma:Inglês
Publicat: 2020
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7184625/
https://ncbi.nlm.nih.gov/pubmed/32208664
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.orglett.0c00885
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