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Improved Stability of Rifampicin in the Presence of Gastric-Resistant Isoniazid Microspheres in Acidic Media

The degradation of rifampicin (RIF) in an acidic medium to form 3-formyl rifamycin SV, a poorly absorbed compound, is accelerated in the presence of isoniazid, contributing to the poor bioavailability of rifampicin. This manuscript presents a novel approach in which isoniazid is formulated into gast...

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Detalhes bibliográficos
Publicado no:Pharmaceutics
Main Authors: Mwila, Chiluba, Walker, Roderick B.
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7150845/
https://ncbi.nlm.nih.gov/pubmed/32151053
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics12030234
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