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Targeting Super‐Enhancers via Nanoparticle‐Facilitated BRD4 and CDK7 Inhibitors Synergistically Suppresses Pancreatic Ductal Adenocarcinoma

Pancreatic ductal adenocarcinoma (PDAC) is a lethal malignant cancer with complex genomic variations, and no targetable genomic lesions have been found yet. Super‐enhancers (SEs) have been found to contribute to the continuous and robust oncogenic transcription. Here, histone H3 lysine 27 acetylatio...

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Detalhes bibliográficos
Publicado no:Adv Sci (Weinh)
Main Authors: Huang, Chen‐Song, You, Xinru, Dai, Chunlei, Xu, Qiong‐Cong, Li, Fuxi, Wang, Li, Huang, Xi‐Tai, Wang, Jie‐Qin, Li, Shi‐Jin, Gao, Zhuoxing, Wu, Jun, Yin, Xiao‐Yu, Zhao, Wei
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7140991/
https://ncbi.nlm.nih.gov/pubmed/32274304
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/advs.201902926
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