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A computational approach yields selective inhibitors of human excitatory amino acid transporter 2 (EAAT2)

Excitatory amino acid transporters (EAATs) represent a protein family that is an emerging drug target with great therapeutic potential for managing central nervous system disorders characterized by dysregulation of glutamatergic neurotransmission. As such, it is of significant interest to discover s...

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Detaylı Bibliyografya
Yayımlandı:J Biol Chem
Asıl Yazarlar: Damm-Ganamet, Kelly L., Rives, Marie-Laure, Wickenden, Alan D., McAllister, Heather M., Mirzadegan, Taraneh
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: American Society for Biochemistry and Molecular Biology 2020
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC7105306/
https://ncbi.nlm.nih.gov/pubmed/32079674
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.AC119.011190
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