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Neurosteroids as Selective Inhibitors of Glycine Receptor Activity: Structure-Activity Relationship Study on Endogenous Androstanes and Androstenes

The ability of androstane and androstene neurosteroids with modifications at C-17, C-5, and C-3 (compounds 1-9) to influence the functional activity of inhibitory glycine and γ-aminobutyric acid (GABA) receptors was estimated. The glycine- and GABA-induced chloride current (I(Gly) and I(GABA)) were...

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Bibliographic Details
Published in:Front Mol Neurosci
Main Authors: Bukanova, Julia V., Solntseva, Elena I., Kudova, Eva
Format: Artigo
Language:Inglês
Published: Frontiers Media S.A. 2020
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Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC7098970/
https://ncbi.nlm.nih.gov/pubmed/32265652
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fnmol.2020.00044
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