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Deubiquitylating enzymes and drug discovery: emerging opportunities
More than a decade after a Nobel Prize was awarded for the discovery of the ubiquitin–proteasome system and clinical approval of proteasome and ubiquitin E3 ligase inhibitors, first-generation deubiquitylating enzyme (DUB) inhibitors are now approaching clinical trials. However, although our knowled...
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| Publicado en: | Nat Rev Drug Discov |
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| Autores principales: | , , , |
| Formato: | Artigo |
| Lenguaje: | Inglês |
| Publicado: |
Nature Publishing Group UK
2017
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| Materias: | |
| Acceso en línea: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7097658/ https://ncbi.nlm.nih.gov/pubmed/28959952 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nrd.2017.152 |
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