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Pharmacokinetic and Pharmacodynamic Considerations for Drugs Binding to Alpha-1-Acid Glycoprotein

According to the free drug hypothesis only the unbound drug is available to act at physiological sites of action, and as such the importance of plasma protein binding primarily resides in its impact on pharmacokinetics and pharmacodynamics. Of the major plasma proteins, alpha-1-acid glycoprotein (AA...

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Dettagli Bibliografici
Pubblicato in:Pharm Res
Autori principali: Smith, Sherri A., Waters, Nigel J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer US 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7089466/
https://ncbi.nlm.nih.gov/pubmed/30593605
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11095-018-2551-x
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