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PROTAC Technology: Opportunities and Challenges

[Image: see text] PROTACs-induced targeted protein degradation has emerged as a novel therapeutic strategy in drug development and attracted the favor of academic institutions, large pharmaceutical enterprises (e.g., AstraZeneca, Bayer, Novartis, Amgen, Pfizer, GlaxoSmithKline, Merck, and Boehringer...

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Pubblicato in:ACS Med Chem Lett
Autori principali: Gao, Hongying, Sun, Xiuyun, Rao, Yu
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2020
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7073876/
https://ncbi.nlm.nih.gov/pubmed/32184950
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.9b00597
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