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Extending the Detection Limit in Fragment Screening of Proteins using Reverse Micelle Encapsulation

Detection of very weak (K(d) > 10 mM) interactions of proteins with small molecules has been elusive. This is particularly important for fragment-based drug discovery where it is suspected that the majority of potentially useful fragments will be invisible to current screening methodologies. We d...

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Pubblicato in:ACS Chem Biol
Autori principali: Fuglestad, Brian, Kerstetter, Nicole E., Bédard, Sabrina, Wand, A. Joshua
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7051832/
https://ncbi.nlm.nih.gov/pubmed/31550881
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.9b00537
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