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Integrating computational lead optimization diagnostics with analog design and candidate selection

AIM: Combining computational lead optimization diagnostics with analog design and computational approaches for assessing optimization efforts are discussed and the compound optimization monitor is introduced. METHODS: Approaches for compound potency prediction are described and a new analog design a...

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Библиографические подробности
Опубликовано в: :Future Sci OA
Главные авторы: Yonchev, Dimitar, Bajorath, Jürgen
Формат: Artigo
Язык:Inglês
Опубликовано: Future Science Ltd 2020
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC7050602/
https://ncbi.nlm.nih.gov/pubmed/32140250
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2144/fsoa-2019-0131
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