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Improvement in predicting drug sensitivity changes associated with protein mutations using a molecular dynamics based alchemical mutation method

While molecular-targeted drugs have demonstrated strong therapeutic efficacy against diverse diseases such as cancer and infection, the appearance of drug resistance associated with genetic variations in individual patients or pathogens has severely limited their clinical efficacy. Therefore, precis...

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Dades bibliogràfiques
Publicat a:Sci Rep
Autors principals: Ono, Fumie, Chiba, Shuntaro, Isaka, Yuta, Matsumoto, Shigeyuki, Ma, Biao, Katayama, Ryohei, Araki, Mitsugu, Okuno, Yasushi
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group UK 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7005789/
https://ncbi.nlm.nih.gov/pubmed/32034220
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-020-58877-9
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