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An Expedient Synthesis of CMF-019: (S)-5-Methyl-3-{1-(pentan-3-yl)-2-(thiophen-2-ylmethyl)-1H-benzo[d]imidazole-5-carboxamido}hexanoic Acid, a Potent Apelin Receptor (APJ) Agonist

BACKGROUND: Apelin receptor (APJ) is a G protein-coupled receptor (GPCR) activated by the endogenous peptide apelin. The apelin–APJ system has emerged as an important regulator of cardiovascular homeostasis. Recently, a potent benzimidazole-derived apelin peptidomimetic, CMF-019, was patented but wi...

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Detalhes bibliográficos
Publicado no:Med Chem
Main Authors: Trifonov, Lena, Afri, Michal, Palczewski, Krzysztof, Korshin, Edward E., Gruzman, Arie
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6993063/
https://ncbi.nlm.nih.gov/pubmed/29651942
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2174/1573406414666180412154952
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