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Hepatic and intestinal biotransformation gene expression and drug disposition in a dextran sulfate sodium-induced colitis mouse model

We examined the impact of gut inflammation on the expression of cytochrome P450 (P450) and other biotransformation genes in male mice using a dextran sulfate sodium (DSS)-induced colitis model. Several P450 isoforms, including CYP1A, CYP2B, CYP2C, and CYP3A, were down-regulated, accompanied by decre...

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Detalhes bibliográficos
Publicado no:Acta Pharm Sin B
Main Authors: Fan, Xiaoyu, Ding, Xinxin, Zhang, Qing-Yu
Formato: Artigo
Idioma:Inglês
Publicado em: Elsevier 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6976992/
https://ncbi.nlm.nih.gov/pubmed/31993311
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.apsb.2019.12.002
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