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Administration of a novel high affinity PICK1 PDZ domain inhibitor attenuates cocaine seeking in rats

Protein interacting with C kinase-1 (PICK1) regulates intra-cellular trafficking of GluA2-containing AMPA receptors, a process known to play a critical role in cocaine-seeking behavior. This suggests that PICK1 may represent a molecular target for developing novel pharmacotherapies to treat cocaine...

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Publicat a:Neuropharmacology
Autors principals: Turner, Christopher, De Luca, Marta, Wolfheimer, Jordan, Hernandez, Nicole, Madsen, Kenneth Lindegaard, Schmidt, Heath D.
Format: Artigo
Idioma:Inglês
Publicat: 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6954965/
https://ncbi.nlm.nih.gov/pubmed/31805281
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuropharm.2019.107901
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