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Toxicity, Pharmacokinetics, and Gut Microbiome of Oral Administration of Sesterterpene MHO7 Derived from a Marine Fungus

Sesterterpene MHO7 derived from mangrove fungus is a novel estrogen receptor degrader for the treatment of breast cancer. To explore its safety and pharmacokinetics in vivo, Log P/D values, stability in simulated gastric/intestinal (SGF/SIF), toxicity, and pharmacokinetics studies were carried mainl...

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Bibliografski detalji
Izdano u:Mar Drugs
Glavni autori: Tian, Wei, Yang, Liang, Wu, Di, Deng, Zixin, Hong, Kui
Format: Artigo
Jezik:Inglês
Izdano: MDPI 2019
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6950057/
https://ncbi.nlm.nih.gov/pubmed/31779201
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/md17120667
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