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Development of Thiazolidinedione-Based HDAC6 Inhibitors to Overcome Methamphetamine Addiction

Thiazolidinedione is a five-membered heterocycle that is widely used in drug discovery endeavors. In this study, we report the design, synthesis, and biological evaluation of a series of thiazolidinedione-based HDAC6 inhibitors. In particular, compound 6b exerts an excellent inhibitory activity agai...

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Detalhes bibliográficos
Publicado no:Int J Mol Sci
Main Authors: Sharma, Chiranjeev, Oh, Yong Jin, Park, Byoungduck, Lee, Sooyeun, Jeong, Chul-Ho, Lee, Sangkil, Seo, Ji Hae, Seo, Young Ho
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6940941/
https://ncbi.nlm.nih.gov/pubmed/31835389
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20246213
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