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Calixmexitil: Calixarene-based Cluster of Mexiletine with Amplified Anti-myotonic Activity as A Novel Use-dependent Sodium Channel Blocker

Mexiletine as the first choice drug in myotonia treatment is a chiral sodium channel blocker clinically used in its racemic form. The phenolic structure of this drug, prompted us to design its novel calix[4]arene-based cluster in a chalice-shaped structure. Therefore, the present study reports the s...

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Pubblicato in:Iran J Pharm Res
Autori principali: Delnavaz Shahr, Amirali, Nasuhi Pur, Fazel
Natura: Artigo
Lingua:Inglês
Pubblicazione: Shaheed Beheshti University of Medical Sciences 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6934949/
https://ncbi.nlm.nih.gov/pubmed/32641945
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.22037/ijpr.2019.1100768
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