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Identifying Promiscuous Compounds with Activity against Different Target Classes

Compounds with multitarget activity are of high interest for polypharmacological drug discovery. Such promiscuous compounds might be active against closely related target proteins from the same family or against distantly related or unrelated targets. Compounds with activity against distinct targets...

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Bibliografski detalji
Izdano u:Molecules
Glavni autori: Feldmann, Christian, Miljković, Filip, Yonchev, Dimitar, Bajorath, Jürgen
Format: Artigo
Jezik:Inglês
Izdano: MDPI 2019
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6891533/
https://ncbi.nlm.nih.gov/pubmed/31752252
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24224185
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