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Natural Product Inspired Novel Indole based Chiral Scaffold Kills Human Malaria Parasites via Ionic Imbalance Mediated Cell Death

Natural products offer an abundant source of diverse novel scaffolds that inspires development of next generation anti-malarials. With this vision, a library of scaffolds inspired by natural biologically active alkaloids was synthesized from chiral bicyclic lactams with steps/scaffold ratio of 1.7:1...

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Dades bibliogràfiques
Publicat a:Sci Rep
Autors principals: Dangi, Poonam, Jain, Ravi, Mamidala, Rajanikanth, Sharma, Vijeta, Agarwal, Shalini, Bathula, Chandramohan, Thirumalachary, M., Sen, Subhabrata, Singh, Shailja
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group UK 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6882913/
https://ncbi.nlm.nih.gov/pubmed/31780808
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-019-54339-z
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