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A Machine Learning-Based Prediction Platform for P-Glycoprotein Modulators and Its Validation by Molecular Docking

P-glycoprotein (P-gp) is an important determinant of multidrug resistance (MDR) because its overexpression is associated with increased efflux of various established chemotherapy drugs in many clinically resistant and refractory tumors. This leads to insufficient therapeutic targeting of tumor popul...

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Publicado en:Cells
Autores principales: Kadioglu, Onat, Efferth, Thomas
Formato: Artigo
Lenguaje:Inglês
Publicado: MDPI 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6829872/
https://ncbi.nlm.nih.gov/pubmed/31640190
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/cells8101286
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