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Continuous Subcutaneous Delivery of Proline-Rich Antimicrobial Peptide Api137 Provides Superior Efficacy to Intravenous Administration in a Mouse Infection Model

Apidaecins are cationic, proline-rich antimicrobial peptides originally isolated from honeybees and exhibit high Gram-negative activity by inhibiting bacterial protein translation. Pharmacokinetics of apidaecin derivative Api137 was studied using single and multiple intravenous or subcutaneous injec...

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Pubblicato in:Front Microbiol
Autori principali: Knappe, Daniel, Schmidt, Rico, Adermann, Knut, Hoffmann, Ralf
Natura: Artigo
Lingua:Inglês
Pubblicazione: Frontiers Media S.A. 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6783563/
https://ncbi.nlm.nih.gov/pubmed/31632382
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fmicb.2019.02283
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