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Tryptoline-Based Benzothiazoles Re-sensitize MRSA to β-Lactam Antibiotics

Resistance-modifying agents (RMAs) offer a promising solution to combat bacterial antibiotic resistance. Here we report the discovery and structure-activity relationships of a new class of RMAs with a novel tryptoline-based benzothiazole scaffold. Our most potent compound in this series (4ad) re-sen...

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Publicado en:Bioorg Med Chem
Autores principales: Wang, Xinfeng, Chen, Jinsen, Wang, Wei, Jaunarajs, Anna, Wang, Xiang
Formato: Artigo
Lenguaje:Inglês
Publicado: 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6779328/
https://ncbi.nlm.nih.gov/pubmed/31521461
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2019.115095
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