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Dual inhibitory action of trazodone on dorsal raphe serotonergic neurons through 5-HT(1A) receptor partial agonism and α(1)-adrenoceptor antagonism

Trazodone is an antidepressant drug with considerable affinity for 5-HT(1A) receptors and α(1)-adrenoceptors for which the drug is competitive agonist and antagonist, respectively. In this study, we used cell-attached or whole-cell patch-clamp recordings to characterize the effects of trazodone at s...

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Publicado en:PLoS One
Autores principales: Montalbano, Alberto, Mlinar, Boris, Bonfiglio, Francesco, Polenzani, Lorenzo, Magnani, Maurizio, Corradetti, Renato
Formato: Artigo
Lenguaje:Inglês
Publicado: Public Library of Science 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6763016/
https://ncbi.nlm.nih.gov/pubmed/31557210
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0222855
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