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Enzyme-Instructed Peptide Assemblies Selectively Inhibit Bone Tumors

Alkaline phosphatases (ALP) contribute to immunosuppression in solid tumors, but they, unfortunately, are “undruggable”. Here we report enzyme-instructed assembly of peptides for selectively inhibiting the tumors that overexpress ALP. We developed a precursor with two parts; an amphiphilic, self-ass...

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Pubblicato in:Chem
Autori principali: Feng, Zhaoqianqi, Han, Xiuguo, Wang, Huaimin, Tang, Tingting, Xu, Bing
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6758912/
https://ncbi.nlm.nih.gov/pubmed/31552305
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chempr.2019.06.020
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