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Multiple Molecular Determinants for Allosteric Modulation of Alternatively Spliced AMPA Receptors

Positive allosteric regulation of glutamate AMPA receptors involves conformational changes that can attenuate receptor desensitization and enhance ion flux through the channel pore. Many allosteric modulators (e.g., cyclothiazide and aniracetam) preferentially affect the flip (i) or flop (o) alterna...

Deskribapen osoa

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Xehetasun bibliografikoak
Argitaratua izan da:J Neurosci
Egile Nagusiak: Quirk, Jennifer C., Nisenbaum, Eric S.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Society for Neuroscience 2003
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6740967/
https://ncbi.nlm.nih.gov/pubmed/14645491
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1523/JNEUROSCI.23-34-10953.2003
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