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Investigation of Dissolution Mechanism and Release Kinetics of Poorly Water-Soluble Tadalafil from Amorphous Solid Dispersions Prepared by Various Methods

The aims of this study were to investigate how the release of tadalafil is influenced by two grades of polyvinylpyrrolidone (Kollidon(®) 12 PF and Kollidon(®) VA 64) and various methods of preparing solid dispersions (solvent evaporation, spray drying and hot-melt extrusion). Tadalafil is poorly wat...

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Publicado en:Pharmaceutics
Autores principales: Školáková, Tereza, Slámová, Michaela, Školáková, Andrea, Kadeřábková, Alena, Patera, Jan, Zámostný, Petr
Formato: Artigo
Lenguaje:Inglês
Publicado: MDPI 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6722951/
https://ncbi.nlm.nih.gov/pubmed/31382377
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics11080383
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