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A Pilot Study towards the Impact of Type 2 Diabetes on the Expression and Activities of Drug Metabolizing Enzymes and Transporters in Human Duodenum

To characterize effects of type 2 diabetes (T2D) on mRNA expression levels for 10 Cytochromes P450 (CYP450s), two carboxylesterases, and three drug transporters (ABCB1, ABCG2, SLCO2B1) in human duodenal biopsies. To compare drug metabolizing enzyme activities of four CYP450 isoenzymes in duodenal bi...

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Detalhes bibliográficos
Publicado no:Int J Mol Sci
Main Authors: Gravel, Sophie, Panzini, Benoit, Belanger, Francois, Turgeon, Jacques, Michaud, Veronique
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6651059/
https://ncbi.nlm.nih.gov/pubmed/31269743
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20133257
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