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Lysosomal P-gp-MDR1 Confers Drug Resistance of Brentuximab Vedotin and Its Cytotoxic Payload Monomethyl Auristatin E in Tumor Cells

Antibody-drug conjugates (ADCs) are composed of an antibody linked to cytotoxic anticancer payloads. ADCs recognize tumor-specific cell surface antigens and are internalized into lysosomes where proteolytic enzymes release the cytotoxic payloads. Efflux transporters on plasma membrane that play a si...

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Detalhes bibliográficos
Publicado no:Front Pharmacol
Main Authors: Liu-Kreyche, Peggy, Shen, Hong, Marino, Anthony M., Iyer, Ramaswamy A., Humphreys, W. Griffith, Lai, Yurong
Formato: Artigo
Idioma:Inglês
Publicado em: Frontiers Media S.A. 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6650582/
https://ncbi.nlm.nih.gov/pubmed/31379564
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fphar.2019.00749
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